| Catalogue number: | PA 14 0081000 |
| Chemical name: | Methylnaltrexone Bromide |
CAS Number: |
73232-52-7 |
| Category: | impurities,metabolites,pharmaceutical standards,intermediates,Fine Chemicals |
| Synonyms: | (17RS)-17-(Cyclopropylmethyl)-4,5α-epoxy-3,14-dihydroxy-17-methyl-6-oxomorphinanium Bromide; N-Methyl Naltrexone Bromide; 17-(Cyclopropylmethyl)-4,5α-epoxy-3,14-dihydroxy-17-methyl-6-oxomorphinanium Bromide; |
| Molecular form: | C21H26BrNO4 |
| Appearance: | White to Pale Brown Solid |
| Mol. Weight: | 436.35 |
| Storage: | 2-8°C Hygroscopic, Refrigerator, Under Inert Atmosphere |
| Shipping Conditions: | Ambient |
| Applications: | A metabolite of Naltrexone. Methylnaltrexone, a selective μ-opioid receptor (MOR) antagonist, functions as a peripherally acting receptor antagonist in tissues of the gastrointestinal tract. When opiates activate μ-opioid receptors (MORs) they trigger signaling pathways that lead to tolerance and hyperalgesia. Methylnaltrexone is positively charged and therefore does not cross the blood brain barier. Mice given morphine with methylnaltrexone experienced pain relief without degeloping tolerance. |
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