Bictegravir-impurities | Pharmaffiliates

Bictegravir and its Impurities

Bictegravir (INN, BIC, formerly known as GS-9883) is an antiviral drug of the integrase inhibitor class that was structurally derived from an earlier compound dolutegravir by scientists at Gilead Sciences. Reference standards of Bictegravir API,and its pharmacopeial, non pharmacopeial impurities, and stable isotopes are listed below.

Displaying 15 results for Bictegravir Impurities
PA 02 1911000

(S)-3,9-Dihydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide

(S)-3,9-Dihydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide


  • Catalogue No.:PA 02 1911000

  • CAS :

    NA

  • Molecular Formula : C21H20F3N3O6

  • Molecular Weight : 467.4

PA 02 1911001

(R)-3,9-Dihydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide

(R)-3,9-Dihydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide


  • Catalogue No.:PA 02 1911001

  • CAS :

    NA

  • Molecular Formula : C21H20F3N3O6

  • Molecular Weight : 467.4

PA 02 1911002

(2R,5S)-8-Hydroxy-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine 6,12-dioxide

(2R,5S)-8-Hydroxy-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine 6,12-dioxide


  • Catalogue No.:PA 02 1911002

  • CAS :

    NA

  • Molecular Formula : C21H18F3N3O7

  • Molecular Weight : 481.38

PA 02 1910000

Bictegravir - API

Bictegravir


  • Catalogue No.:PA 02 1910000

  • CAS :

    1611493-60-7

  • Molecular Formula : C21H18F3N3O5

  • Molecular Weight : 449.39

PA 02 1911003

(2S,5R,13aS)-8-Hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

(2S,5R,13aS)-8-Hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide


  • Catalogue No.:PA 02 1911003

  • CAS :

    1616340-12-5

  • Molecular Formula : C21H18F3N3O5

  • Molecular Weight : 449.39

PA 02 1911004

(2R,5R,13aR)-8-Hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

(2R,5R,13aR)-8-Hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide


  • Catalogue No.:PA 02 1911004

  • CAS :

    1846582-14-6

  • Molecular Formula : C21H18F3N3O5

  • Molecular Weight : 449.39

PA 02 1911005

(2R,5S,13aR)-8-Methoxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

(2R,5S,13aR)-8-Methoxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide


  • Catalogue No.:PA 02 1911005

  • CAS :

    1616340-94-3

  • Molecular Formula : C22H20F3N3O5

  • Molecular Weight : 463.41

PA 02 1911006

(2R,5S,13aR)-N-(2,4-Difluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

(2R,5S,13aR)-N-(2,4-Difluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide


  • Catalogue No.:PA 02 1911006

  • CAS :

    1611493-56-1

  • Molecular Formula : C21H19F2N3O5

  • Molecular Weight : 431.4

PA 02 1911007

(2S,5R,13aS)-N-(2-Fluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

(2S,5R,13aS)-N-(2-Fluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide


  • Catalogue No.:PA 02 1911007

  • CAS :

    1616339-90-2

  • Molecular Formula : C21H20FN3O5

  • Molecular Weight : 413.41

PA 02 1911008

(2S,5R,13aS)-N-(4-Fluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

(2S,5R,13aS)-N-(4-Fluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide


  • Catalogue No.:PA 02 1911008

  • CAS :

    1616339-82-2

  • Molecular Formula : C21H20FN3O5

  • Molecular Weight : 413.41

PA 02 1911009

(2S,5R,13aS)-N-(2,6-Difluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

(2S,5R,13aS)-N-(2,6-Difluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide


  • Catalogue No.:PA 02 1911009

  • CAS :

    1616340-13-6

  • Molecular Formula : C21H19F2N3O5

  • Molecular Weight : 431.4

PA 02 1911010

Methyl 5-acetyl-1-(2,2-dimethoxyethyl)-3-methoxy-4-oxo-1,4-dihydropyridine-2-carboxylate

Methyl 5-acetyl-1-(2,2-dimethoxyethyl)-3-methoxy-4-oxo-1,4-dihydropyridine-2-carboxylate


  • Catalogue No.:PA 02 1911010

  • CAS :

    1335210-23-5

  • Molecular Formula : C14H19NO7

  • Molecular Weight : 313.31

PA 02 1911011

(2S,3S,4S,5R,6S)-6-(((2R,5S,13aR)-7,9-Dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepin-8-yl)oxy)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylic acid

(2S,3S,4S,5R,6S)-6-(((2R,5S,13aR)-7,9-Dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepin-8-yl)oxy)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylic acid


  • Catalogue No.:PA 02 1911011

  • CAS :

    2365156-60-9

  • Molecular Formula : C27H26F3N3O11

  • Molecular Weight : 625.51

PA STI 089238

Bictegravir-13C-15N-d2

Bictegravir-13C-15N-d2


  • Catalogue No.:PA STI 089238

  • CAS :

    NA

  • Molecular Formula : C2013CH16D2F3N215NO5

  • Molecular Weight : 453.38

PA 02 1911012

9-Hydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,8-dihydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide

9-Hydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,8-dihydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide


  • Catalogue No.:PA 02 1911012

  • CAS :

    NA

  • Molecular Formula : C21H18F3N3O5

  • Molecular Weight : 449.39