Bictegravir

Bictegravir (INN, BIC, formerly known as GS-9883) is an antiviral drug of the integrase inhibitor class that was structurally derived from an earlier compound dolutegravir by scientists at Gilead Sciences. Reference standards of Bictegravir API,and its pharmacopeial, non pharmacopeial impurities, and stable isotopes are listed below.

stdClass Object
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    [pname] => (S)-3,9-Dihydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide
    [catalogue_number] => PA 02 1911000
    [category_ids] => ,78,75,70,76,82,
    [chemical_name] => 
    [weight] => 467.4
    [form] => C21H20F3N3O6
    [cas] => NA
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PA 02 1911000

(S)-3,9-Dihydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide

  • Catalogue No.:PA 02 1911000

  • CAS :

    NA

  • Molecular Formula : C21H20F3N3O6

  • Molecular Weight : 467.4

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Details 
stdClass Object
(
    [pname] => (R)-3,9-Dihydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide
    [catalogue_number] => PA 02 1911001
    [category_ids] => ,78,75,70,76,82,
    [chemical_name] => 
    [weight] => 467.4
    [form] => C21H20F3N3O6
    [cas] => NA
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PA 02 1911001

(R)-3,9-Dihydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide

  • Catalogue No.:PA 02 1911001

  • CAS :

    NA

  • Molecular Formula : C21H20F3N3O6

  • Molecular Weight : 467.4

Enquire
Details 
stdClass Object
(
    [pname] => (2R,5S)-8-Hydroxy-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine 6,12-dioxide
    [catalogue_number] => PA 02 1911002
    [category_ids] => ,78,75,70,76,82,
    [chemical_name] => 
    [weight] => 481.38
    [form] => C21H18F3N3O7
    [cas] => NA
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PA 02 1911002

(2R,5S)-8-Hydroxy-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine 6,12-dioxide

  • Catalogue No.:PA 02 1911002

  • CAS :

    NA

  • Molecular Formula : C21H18F3N3O7

  • Molecular Weight : 481.38

Enquire
Details 
stdClass Object
(
    [pname] => (2S,5R,13aS)-8-Hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
    [catalogue_number] => PA 02 1911003
    [category_ids] => ,75,76,78,70,82,
    [chemical_name] => 
    [weight] => 449.39
    [form] => C21H18F3N3O5
    [cas] => 1616340-12-5
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PA 02 1911003

(2S,5R,13aS)-8-Hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

  • Catalogue No.:PA 02 1911003

  • CAS :

    1616340-12-5

  • Molecular Formula : C21H18F3N3O5

  • Molecular Weight : 449.39

Enquire
Details 
stdClass Object
(
    [pname] => (2R,5R,13aR)-8-Hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
    [catalogue_number] => PA 02 1911004
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    [chemical_name] => 
    [weight] => 449.39
    [form] => C21H18F3N3O5
    [cas] => 1846582-14-6
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PA 02 1911004

(2R,5R,13aR)-8-Hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

  • Catalogue No.:PA 02 1911004

  • CAS :

    1846582-14-6

  • Molecular Formula : C21H18F3N3O5

  • Molecular Weight : 449.39

Enquire
Details 
stdClass Object
(
    [pname] => (2R,5S,13aR)-8-Methoxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
    [catalogue_number] => PA 02 1911005
    [category_ids] => ,75,76,78,70,82,
    [chemical_name] => 
    [weight] => 463.41
    [form] => C22H20F3N3O5
    [cas] => 1616340-94-3
    [pslug] => 1616340-94-3-2r-5s-13ar-8-methoxy-7-9-dioxo-n-2-4-6-trifluorobenzyl-2-3-4-5-7-9-13-13a-octahydro-2-5-methanopyrido-1-2-4-5-pyrazino-2-1-b-1-3-oxazepine-10-carboxamide-pa021911005
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PA 02 1911005

(2R,5S,13aR)-8-Methoxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

  • Catalogue No.:PA 02 1911005

  • CAS :

    1616340-94-3

  • Molecular Formula : C22H20F3N3O5

  • Molecular Weight : 463.41

Enquire
Details 
stdClass Object
(
    [pname] => (2R,5S,13aR)-N-(2,4-Difluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
    [catalogue_number] => PA 02 1911006
    [category_ids] => ,75,76,78,70,82,
    [chemical_name] => 
    [weight] => 431.4
    [form] => C21H19F2N3O5
    [cas] => 1611493-56-1
    [pslug] => 1611493-56-1-2r-5s-13ar-n-2-4-difluorobenzyl-8-hydroxy-7-9-dioxo-2-3-4-5-7-9-13-13a-octahydro-2-5-methanopyrido-1-2-4-5-pyrazino-2-1-b-1-3-oxazepine-10-carboxamide-pa021911006
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PA 02 1911006

(2R,5S,13aR)-N-(2,4-Difluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

  • Catalogue No.:PA 02 1911006

  • CAS :

    1611493-56-1

  • Molecular Formula : C21H19F2N3O5

  • Molecular Weight : 431.4

Enquire
Details 
stdClass Object
(
    [pname] => (2S,5R,13aS)-N-(2-Fluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
    [catalogue_number] => PA 02 1911007
    [category_ids] => ,75,76,78,70,82,
    [chemical_name] => 
    [weight] => 413.41
    [form] => C21H20FN3O5
    [cas] => 1616339-90-2
    [pslug] => 1616339-90-2-2s-5r-13as-n-2-fluorobenzyl-8-hydroxy-7-9-dioxo-2-3-4-5-7-9-13-13a-octahydro-2-5-methanopyrido-1-2-4-5-pyrazino-2-1-b-1-3-oxazepine-10-carboxamide-pa021911007
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PA 02 1911007

(2S,5R,13aS)-N-(2-Fluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

  • Catalogue No.:PA 02 1911007

  • CAS :

    1616339-90-2

  • Molecular Formula : C21H20FN3O5

  • Molecular Weight : 413.41

Enquire
Details 
stdClass Object
(
    [pname] => (2S,5R,13aS)-N-(4-Fluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
    [catalogue_number] => PA 02 1911008
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    [chemical_name] => 
    [weight] => 413.41
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PA 02 1911008

(2S,5R,13aS)-N-(4-Fluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

  • Catalogue No.:PA 02 1911008

  • CAS :

    1616339-82-2

  • Molecular Formula : C21H20FN3O5

  • Molecular Weight : 413.41

Enquire
Details 
stdClass Object
(
    [pname] => (2S,5R,13aS)-N-(2,6-Difluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
    [catalogue_number] => PA 02 1911009
    [category_ids] => ,75,76,78,70,82,
    [chemical_name] => 
    [weight] => 431.4
    [form] => C21H19F2N3O5
    [cas] => 1616340-13-6
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PA 02 1911009

(2S,5R,13aS)-N-(2,6-Difluorobenzyl)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide

  • Catalogue No.:PA 02 1911009

  • CAS :

    1616340-13-6

  • Molecular Formula : C21H19F2N3O5

  • Molecular Weight : 431.4

Enquire
Details 
stdClass Object
(
    [pname] => (2S,3S,4S,5R,6S)-6-(((2R,5S,13aR)-7,9-Dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepin-8-yl)oxy)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylic acid
    [catalogue_number] => PA 02 1911011
    [category_ids] => ,75,76,78,70,82,
    [chemical_name] => 
    [weight] => 625.51
    [form] => C27H26F3N3O11
    [cas] => 2365156-60-9
    [pslug] => 2365156-60-9-2s-3s-4s-5r-6s-6-2r-5s-13ar-7-9-dioxo-10-2-4-6-trifluorobenzyl-carbamoyl-2-3-4-5-7-9-13-13a-octahydro-2-5-methanopyrido-1-2-4-5-pyrazino-2-1-b-1-3-oxazepin-8-yl-oxy-3-4-5-trihydroxytetrahydro-2h-pyran-2-carboxylic-acid-pa021911011
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PA 02 1911011

(2S,3S,4S,5R,6S)-6-(((2R,5S,13aR)-7,9-Dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepin-8-yl)oxy)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylic acid

  • Catalogue No.:PA 02 1911011

  • CAS :

    2365156-60-9

  • Molecular Formula : C27H26F3N3O11

  • Molecular Weight : 625.51

Enquire
Details 
stdClass Object
(
    [pname] => Bictegravir-13C-15N-d2
    [catalogue_number] => PA STI 089238
    [category_ids] => ,98,75,76,78,70,82,
    [chemical_name] => 
    [weight] => 453.38
    [form] => C2013CH16D2F3N215NO5
    [cas] => NA
    [pslug] => bictegravir-13c-15n-d2-pasti089238
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PA STI 089238

Bictegravir-13C-15N-d2

  • Catalogue No.:PA STI 089238

  • CAS :

    NA

  • Molecular Formula : C2013CH16D2F3N215NO5

  • Molecular Weight : 453.38

Enquire
Details 
stdClass Object
(
    [pname] => 9-Hydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,8-dihydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide
    [catalogue_number] => PA 02 1911012
    [category_ids] => ,75,76,78,70,82,
    [chemical_name] => 
    [weight] => 449.39
    [form] => C21H18F3N3O5
    [cas] => NA
    [pslug] => 9-hydroxy-2-1s-3r-3-hydroxycyclopentyl-1-8-dioxo-n-2-4-6-trifluorobenzyl-1-8-dihydro-2h-pyrido-1-2-a-pyrazine-7-carboxamide-pa021911012
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PA 02 1911012

9-Hydroxy-2-((1S,3R)-3-hydroxycyclopentyl)-1,8-dioxo-N-(2,4,6-trifluorobenzyl)-1,8-dihydro-2H-pyrido[1,2-a]pyrazine-7-carboxamide

  • Catalogue No.:PA 02 1911012

  • CAS :

    NA

  • Molecular Formula : C21H18F3N3O5

  • Molecular Weight : 449.39

Enquire
Details 
stdClass Object
(
    [pname] => (2R,5S,13aR)-8-Hydroxy-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine 6,12-dioxide
    [catalogue_number] => PA 02 1911013
    [category_ids] => ,78,75,70,76,82,
    [chemical_name] => 
    [weight] => 481.38
    [form] => C21H18F3N3O7
    [cas] => NA
    [pslug] => 2r-5s-13ar-8-hydroxy-7-9-dioxo-10-2-4-6-trifluorobenzyl-carbamoyl-2-3-4-5-7-9-13-13a-octahydro-2-5-methanopyrido-1-2-4-5-pyrazino-2-1-b-1-3-oxazepine-6-12-dioxide-pa021911013
    [latest_product] => 0
    [linkproducts] => 0
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PA 02 1911013

(2R,5S,13aR)-8-Hydroxy-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine 6,12-dioxide

  • Catalogue No.:PA 02 1911013

  • CAS :

    NA

  • Molecular Formula : C21H18F3N3O7

  • Molecular Weight : 481.38

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CPHI INDIA- 28, 30 November